Nermin Samir

nerminsamir@pharma.asu.edu.eg

Internal ID: rp13390

Publications

Results 1-18 of 18 (Search time: 0.0 seconds).

Issue DateTitleAuthor(s)
12026Towards the discovery of potent epigenetic modulators: Design, synthesis, biological evaluation, and SAR investigation of novel indole-based derivatives targeting HDAC1 and HDAC6Shawky, Sarah; Ahmed, Tarek Erfan; Haffez, Hesham; Sobhy, Aya; Soror, Sameh; Jaballah, Maiy; Henary, Maged; Nermin Samir ; Lasheen, Deena S
22025Novel isatin conjugates endowed with analgesic and anti-inflammatory properties: design, synthesis and biological evaluationBrown, LaVauria D; Girgis, Adel S; Patel, Shruti; Said, Mona F; Baidya, Anurag TK; Kumar, Rajnish; Moore, Jade; Khadanga, Anshuman; Sakhuja, Rajeev; Nermin Samir 
32025Chalcones Tethered with Pyridylmethyloxy Tail: Unlocking New Pathways in MDM2-p53 Targeted Cancer TreatmentAlnaeb, Suha; Jaballah, Maiy Y; Morsy, Mohamed A; Abouzid, Khaled AM; Nermin Samir ; Adel, Mai
42025Next-Generation Diarylurea Antibacterials: From Structural Design and Optimization to Microbial Target Specific StrategiesKassab, Rafif Rashad; Serya, Rabah Ahmed; Serya, Rabah ; Nermin Samir ; Abouzid, Khaled
52025The recent advances in benzimidazole-based antimicrobials and antitubercular agentsTarek, Abdalrahman; Jaballah, Maiy Y; Elrazaz, Eman Z; Nermin Samir 
62024Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: Design, synthesis and anti-proliferative activityHigazy, Samah; El-Khouly, Ahmed; Giovannuzzi, Simone; Begines, Paloma; Gaber, Hatem M; Supuran, Claudiu T; Abouzid, Khaled AM; Nermin Samir 
72024Design, synthesis and molecular modeling of Pyrazolo [1, 5-a] pyrimidine derivatives as dual inhibitors of CDK2 and TRKA kinases with Antiproliferative activityAttia, Mohamed H; Taher, Azza T; Abdel-Aziz, Hatem A; Abou El Ella, Dalal A; Nermin Samir ; Lasheen, Deena S
82024Targeting apoptosis; design, synthesis and biological evaluation of new benzoxazole and thiazole based derivativesHelmy, Sama W; Ella, Dalal A Abou El; Nermin Samir ; Shahin, Mai I; Lasheen, Deena S
92023New NSAID conjugates as potent and selective COX-2 inhibitors: synthesis, molecular modeling and biological investigationBokhtia, Riham M; Panda, Siva S; Girgis, Adel S; Said, Mona F; Abdelnaser, Anwar; Nasr, Soad; Bekheit, Mohamed S; Dawood, Abdelhameed S; Sharma, Horrick; Nermin Samir 
102023Design, synthesis, and biological evaluation with molecular dynamics study of novel pyrazolo [3, 4-d] pyrimidine derivatives as anti-cancer agentsShaban, Rania M; Nissan, Yassin M; Abouzid, Khaled AM; Nermin Samir 
112022Design and synthesis of ibuprofen-quinoline conjugates as potential anti-inflammatory and analgesic drug candidatesGhanim, Amany M; Girgis, Adel S; Kariuki, Benson M; Said, Mona F; Abdelnaser, Anwar; Nasr, Soad; Bekheit, Mohamed S; Abdelhameed, Mohamed F; Almalki, Ahmad J; Nermin Samir 
122022A fluorescence-based assay to probe inhibitory effect of Fructose mimics on GLUT5 transport in breast Cancer cellsRana, Natasha; Aziz, Marwa A; Wuest, Frank; Abouzid, Khaled AM; West, FG; Nermin Samir ; Serya, Rabah AT; Lasheen, Deena S
1318-Aug-2020Design, Synthesis, and Biological Evaluation of Novel 7H-[1,2,4]Triazolo[3,4-b][1,3,4]thiadiazine Inhibitors as Antitumor AgentsIsmail, Muhammad I; Mohamady, Samy; Abouzid, Khaled ; Nermin Samir 
142020Synthesis of some tropane-based compounds targeting colon cancerGeorge, Riham F; Elrazaz, Eman ; Ayoub, Iriny M; Shalaby, ElSayed M; Plaisier, Jasper R; Demitri, Nicola; Wink, Michael; Nermin Samir 
152020Molecular dynamic study and synthesis of 1H-benzo [d] imidazole-5-carboxamide derivatives as inhibitors for yellow fever and zika virus replicationMitry, Madonna; El-Araby, Amr; Neyts, Johan; Kaptein, Suzanne; Nermin Samir ; Serya, Rabah AT
162018HIV-1 RT-Associated RNase H reviewMitry, Madonna; Abdou, Nermin S; Nermin Samir ; Serya, Rabah AT
172018Synthesis, antiproliferative activity and 2D-QSAR study of some 8-alkyl-2, 4-bisbenzylidene-3-nortropinonesGeorge, Riham F; Ayoub, Iriny M; Shalaby, ElSayed M; Demitri, Nicola; Wink, Michael; Nermin Samir 
182017An overview on the prospective CDKs inhibitors as anti-cancer drugsOudah, Khulood H; Serya, R; Abouzid, K; Serya, Rabah ; Nermin Samir