Name
Bioorganic Chemistry
ISSN
0045-2068

Puplications
(All)

Results 21-40 of 40 (Search time: 0.0 seconds).

Issue DateTitleAuthor(s)
21Jun-2014Molecular design and synthesis of 1,4-disubstituted piperazines as α(1)-adrenergic receptor blockersHussein, Mohammed M; Serya, Rabah ; Abdel Naby, Rana M; Al-Abd, Ahmed M; Saleh, Dalia O; El-Eraky, Wafaa I; Khaled A M Abouzid ; Abou El Ella, Dalal 
22026Multitarget bioactive benzo [f] quinoline heterocycles from a thiocarbohydrazone scaffold: synthesis, biological assays, and in silico mechanistic rationaleSaleh, Esraa M; El-Banna, Mohamed G; Fahim, Asmaa M; El Awady, Mohamed E; Rizk, Sameh A; Eman A. E. El-Helw 
316-Jul-2021New N-(1,3,4-thiadiazol-2-yl)furan-2-carboxamide derivatives as potential inhibitors of the VEGFR-2Soliman Farag Saad, Paula ; Hemdan, Magdy M. ; El-Sayed, Wael ; Mohamed Hussein Hussein Moustafa Hekal 
4Apr-2023New trends in synthetic drugs and natural products targeting 20S proteasomes in cancersAtta, Hind; Alzahaby, Nouran ; Hamdy, Nadia M; Emam, Soha H; Sonousi, Amr; Ziko, Laila
5Dec-2022Novel 1,3-diaryl pyrazole derivatives bearing methylsulfonyl moiety: Design, synthesis, molecular docking and dynamics, with dual activities as anti-inflammatory and anticancer agents through selectively targeting COX-2Shaker, Ahmed M M; Shahin, Mai I. ; AboulMagd, Asmaa M; Abdel Aleem, Seham A; Abdel-Rahman, Hamdy M; Abou El Ella, Dalal 
62022Novel Azine Linked Hybrids of 2-Indolinone and Thiazolodinone Scaffolds as CDK2 Inhibitors with Potential Anticancer Activity: In Silico Design, Synthesis, Biological, Molecular Dynamics and Binding Free Energy StudiesQayed, Wesam S; Hassan, Mostafa A; El-Sayed, Wael ; Rogério A Silva, José; Aboul-Fadl, Tarek 
71-Feb-2024Novel indolinone-tethered benzothiophenes as anti-tubercular agents against MDR/XDR M. tuberculosis: Design, synthesis, biological evaluation and in vivo pharmacokinetic studyEldehna, Wagdy M.; Mahmoud, Sally Tarek; Elshnawey, Esraa R.; Elsayed, Zainab M.; Majrashi, Taghreed A.; El-Ashrey, Mohamed K.; Rashed, Mahmoud; Hemeda, Loah R.; Shoun, Aly A.; Elkaeed, Eslam B.; El Hassab, Mahmoud A.; Abdel-Aziz, Marwa M.; Shahin, Mai I. 
81-Dec-2017Novel quinoline-3-carboxamides (Part 2): Design, optimization and synthesis of quinoline based scaffold as EGFR inhibitors with potent anticancer activityAly, Rasha M.; Serya, Rabah ; El-Motwally, Amira M.; Abbas, Safinaz; Abou El Ella, Dalal ; Esmat, Ahmed 
9Aug-2020Scaffold hopping and redesign approaches for quinazoline based urea derivatives as potent VEGFR-2 inhibitorsHadi, Soha R Abd El; Soliman, Dalia H; Elrazaz, Eman ; Khaled A M Abouzid ; Lasheen, Deena S. 
1029-Sep-2025Straightforward synthesis and in silico evaluation of pyrazolylthiazolidinone derivatives as prospective antiproliferative agentsRamadan, Sayed ; Gomha, Sobhi M; El-Helw, Eman A. E. 
11Oct-2025Straightforward synthesis and in silico evaluation of pyrazolylthiazolidinone derivatives as prospective antiproliferative agentsRamadan, Sayed K. ; Gomha, Sobhi M; Eman A. E. El-Helw 
12Feb-2022Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activityRagab, Mahmoud A; Elagawany, Mohamed; Daabees, Hoda; Ahmed, Al-Shaimaa F; Awad, Eman M; Billon, Cyrielle; Elgendy, Bahaa; Abouzid, Khaled ; Kassab, Shaymaa E
13Jan-2020Synthesis and antimicrobial evaluation of new halogenated 1,3-Thiazolidin-4-onesHammad, Shaymaa G; El-Gazzar, Marwa G; Abutaleb, Nader S; Li, Daoyi; Ramming, Isabell; Shekhar, Aditya; Abdel-Halim, Mohammad; Elrazaz, Eman ; Seleem, Mohamed N; Bilitewski, Ursula; El-Hossary, Ebaa M; Khaled A M Abouzid 
142026Synthesis and biological evaluation of novel heterocyclic compounds derived from ammonium thiocyanate for control of Culex pipiens and Musca domestica.Ghareeb, Eman A; Kamal, Mahmoud; Farag, Shaimaa M; Ammar, Asmaa M; Mahmoud, Naglaa FH; Eman A. E. El-Helw 
15Jul-2021Synthesis, DFT, and eco-friendly insecticidal activity of some N-heterocycles derived from 4-((2-oxo-1,2-dihydroquinolin-3-yl)methylene)-2-phenyloxazol-5(4H)-oneGhareeb, Eman A; Mahmoud, Naglaa F H; El-Bordany, Eman A; El-Helw, EAE 
16Sep-2021Synthesis, in vitro biological investigation, and molecular dynamics simulations of thiazolopyrimidine based compounds as corticotrophin releasing factor receptor-1 antagonistsElgiushy, Hossam R; Abou-Taleb, Nageh A; Holz, George G; Chepurny, Oleg G; Pirmettis, Ioannis; Kakabakos, Sotirios; Karageorgos, Vlasios; Liapakis, George; Albohy, Amgad; Abouzid, Khaled ; Hammad, Sherif F
1727-Dec-2024Synthesis, in vivo evaluation, and in silico molecular docking of benzo[h]quinoline derivatives as potential Culex pipiens L. larvicidesRamadan, Sayed ; Hosni, Eslam M; Kamal, Mahmoud ; El-Helw, Eman A. E. ; Hashem, Ahmed ; Wael Abou-Elmagd 
182024Synthesis, insecticidal Activity, and molecular docking analysis of some benzo[h]quinoline derivatives against Culex pipiens L. LarvaeHosni, Eslam M.; Mahmoud Kamal ; Sayed Karam Ramadan Emam ; Eman A.E. El-Helw ; Hashem, Ahmed 
192023Synthesis, larvicidal efficiency and molecular docking studies of novel annulated pyrano [2, 3-c] pyrazoles against Culex pipiens L. and Musca domestica L. larvaeEl-Sayed, Mahmoud KF; El-Shahawi, Manal M; Ali, Yasmeen M; El-Azm, Fatma SM Abu; Doaa Ramadan Abdel Haleem Ramadan ; M.M Elshahawi, Manal M. Elshahawi, Manal Mohamed El-Shahawi, Manal M. El-Shahawi 
201-Dec-2024Unveiling the anticancer potential of novel spirooxindole-tethered pyrazolopyridine derivativesEldehna, Wagdy M.; Abdulla, Maha Hamadien; Nafie, Mohamed S.; Elsawi, Ahmed E.; Ayman, Salsabil; Shahin, Mai I. ; Alhassan, Noura S.; Zubaidi, Ahmad M.; Ghabbour, Hazem A.; Elaasser, Mahmoud; Al-Karmalawy, Ahmed A.; Abdel-Aziz, Hatem A.