Department of Pharmaceutical Chemistry - Pharmacy

Cairo, Abbassia, EG

OrgUnit's Researchers publications
(Dept/Workgroup Publication)

Results 141-160 of 199 (Search time: 0.0 seconds).

Issue DateTitleAuthor(s)
1412016Pyrazolo[3,4-d]pyrimidine based scaffold derivatives targeting kinases as anticancer agentsIsmail, Nasser S.M.; Ali, Eslam M.H.; Ibrahim, Diaa A.; Serya, Rabah A.T. ; Abou El Ella, Dalal 
2Mar-2017Pyridazine Based Scaffolds as Privileged Structures in anti-Cancer TherapyJaballah, Maiy Youssef; Serya, Rabah Taha; Abouzid, Khaled 
31-Jan-2008Pyridazinone derivatives: design, synthesis, and in vitro vasorelaxant activityAbouzid, Khaled ; Abdel Hakeem, Maha; Khalil, Omnya; Maklad, Yosria
416-Aug-2024Pyridazinone-based derivatives as anticancer agents endowed with anti-microbial activity: molecular design, synthesis, and biological investigationEl-Nagar, Mohamed K.S.; Shahin, Mai I. ; El-Behairy, Mohammed F.; Taher, Ehab S.; El-Badawy, Mohamed F.; Sharaky, Marwa; Abou El Ella, Dalal A.; Abouzid, Khaled A.M.; Adel, Mai
5Sep-2018Pyrrolopyrimidine, A Multifaceted Scaffold in Cancer Targeted TherapyAdel, Mai; Serya, Rabah A T ; Lasheen, Deena S. ; Abouzid, Khaled 
61-Aug-2013Quinazoline and tetrahydropyridothieno[2,3-d]pyrimidine derivatives as irreversible EGFR tyrosine kinase inhibitors: Influence of the position 4 substituentHamed, Mostafa M.; Abou El Ella, Dalal ; Keeton, Adam B.; Piazza, Gary A.; Engel, Matthias; Hartmann, Rolf W.; Abadi, Ashraf H.
7May-2016Quinoline-based small molecules as effective protein kinases inhibitors (Review)Rasha M. Aly; Rabah A. T. Serya; Amira M. El-Motwally; Ghada H. Al-Ansary; Abou El Ella, Dalal 
8May-2016Quinoxaline-Based Scaffolds Targeting Tyrosine Kinases and Their Potential Anticancer ActivityEl Newahie, Aliya M S; Ismail, Nasser S M; Abou El Ella, Dalal ; Abouzid, Khaled 
92015Radioiodination and biological evaluation of Cladribine as potential agent for tumor imaging and therapyBayoumi, NA; Amin, AM; Ismail, NSM; Abouzid, Khaled ; El-Kolaly, MT
1022-Dec-2022SAR investigation and optimization of benzimidazole-based derivatives as antimicrobial agents against Gram-negative bacteriaDokla, Eman ; Abutaleb, Nader S; Milik, Sandra N; Kandil, Ezzat A E A; Qassem, Omar M; Elgammal, Yehia; Nasr, Maha ; McPhillie, Martin J; Abouzid, Khaled A M; Seleem, Mohamed N; Imming, Peter; Adel, Mai
11Aug-2020Scaffold hopping and redesign approaches for quinazoline based urea derivatives as potent VEGFR-2 inhibitorsHadi, Soha R Abd El; Soliman, Dalia H; Elrazaz, Eman ; Khaled A M Abouzid ; Lasheen, Deena S. 
12May-2025Structural Optimization and MD Simulation Study of Benzimidazole Derivatives as Potent Mutant FLT3 Kinase Inhibitors Targeting AMLEl-Deen, Nada Alaa; DeFilippis, RosaAnna; Milik, Sandra N; Patel, Suhana; Ismail, Muhammad I; Khaled, Omar; Ahmed, Tarek Erfan; Abdelfattah, Ayatullah Gamal; Ali, Eslam M H; Gaballah, Maiy Y; McPhillie, Martin J; Abouzid, Khaled A M; Henary, Maged; Minucci, Saverio; Shah, Neil P; Abdel-Aziz, Amal Kamal ; Serya, Rabah ; Dokla, Eman 
13Apr-2021Structure- and Ligand-Based in silico Studies towards the Repurposing of Marine Bioactive Compounds to Target SARS-CoV-2Fayed, Marwa A A; El-Behairy, Mohammed Farrag; Abdallah, Inas A; Abdel-Bar, Hend Mohamed; Elimam, Hanan; Mostafa, Ahmed; Moatasim, Yassmin; Abouzid, Khaled ; Elshaier, Yaseen A M M
14Feb-2022Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activityRagab, Mahmoud A; Elagawany, Mohamed; Daabees, Hoda; Ahmed, Al-Shaimaa F; Awad, Eman M; Billon, Cyrielle; Elgendy, Bahaa; Abouzid, Khaled ; Kassab, Shaymaa E
15Mar-2013Structure-based design and synthesis of novel pseudosaccharine derivatives as antiproliferative agents and kinase inhibitorsElsayed, Mohamed S A; El-Araby, Moustafa E; Serya, Rabah ; El-Khatib, Ahmed H; Linscheid, Michael W; Khaled A M Abouzid 
162010Structure-based molecular design, synthesis, and in vivo anti-inflammatory activity of pyridazinone derivatives as nonclassic COX-2 inhibitorsAbouzid, Khaled ; Khalil, NA; Ahmed, E.M. ; El-Latif, HAA; El-Araby, ME
171999Substrate specificity and stereoselectivity of rat brain microsomal anandamide amidohydrolaseLang, WS; Qin, C; Lin, SY; Khanolkar, AD; Goutopoulos, A; Fan, PS; Abouzid, Khaled ; Meng, ZX; Biegel, D; Makriyannis, A
1815-Jul-2018Surmounting the resistance against EGFR inhibitors through the development of thieno[2,3-d]pyrimidine-based dual EGFR/HER2 inhibitorsMilik, Sandra N; Serya, Rabah ; Minucci, Saverio; Lasheen, Deena S. ; Khaled A M Abouzid ; Abdel-Aziz, Amal Kamal 
19Aug-2012Synthesis and anti-proliferative activity of substituted-anilinoquinazolines and its relation to EGFR inhibitionEl Ella, D A A; Saleh, K A; Hassan, M; El-Araby, M E; Abouzid, Khaled ; Prof. Hamdy, Nadia M. 
20Oct-2013Synthesis and Antifungal Activity of Some New Substituted5, 7- Diiodo-8-Hydroxy Quinoline DerivativesHoda H. Fahmy; Nagy M. Khalifa; Abou El Ella, Dalal ; Mohamed A. Ismail; Noha M. Mostafa; Abdelhamid A. Hamdy